生物活性
CAY10603是一种强效的选择性HDAC6抑制剂,IC50为2 pM,选择性比其它HDACs高200多倍。
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体外研究
CAY10603, via inhibition of HDAC6, shows potent antiproliferative activity against pancreatic cancer cell lines with IC50 of <1 μM, which can be used as a new molecular probe in exploring HDAC biology.
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