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CAS-Nr. | 76530-44-4 |
Bezeichnung: | |
Englisch Name: | Azamulin |
Synonyma: | Azamulin;SA 85530b;TMD 85-530, SA 85530b;Antibiotic TDM 85-530;14-O-(5-(2-Amino1,3,4-triazolyl)thioacetyl)dihydromutilin;[(5-Amino-1H-1,2,4-triazol-3-yl)thio]acetic acid (3aS,4R,5S,6R,8R,9R,9aR,10R)-6-ethyldecahydro-5-hydroxy-4,6,9,10-tetramethyl-1-oxo-3a,9-propano-3aH-cyclopentacycloocten-8-yl ester |
CBNumber: | CB51176138 |
Summenformel: | C24H38N4O4S |
Molgewicht: | 0 |
MOL-Datei: | 76530-44-4.mol |
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Azamulin physikalisch-chemischer Eigenschaften |
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storage temp. : |
-20°C Freezer |
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Stabilität:: |
Store at -200C. |
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Azamulin Chemische Eigenschaften,Einsatz,Produktion Methoden |
Chemische Eigenschaften White Solid |
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Verwenden Azamulin is a semi-synthetic pleuromutilin prepared by sequential reaction of dihydropleuromutilin tosylate with 2-amino-1,2,4-triazole-5-thiol. While azamulin is a broad spectrum antibiotic in the pleuromutilin class, this aspect of its bioprofile has received little attention. In fact, the triazole substituent added to nominally improve the drugs bioavailability, imparted an unusual selectivity for the inhibition of specific cytochrome P450 mixed function oxidase sub-types, important for understanding the manner in which the body metabolises drugs or xenobiotics. |
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Verwenden It is a highly selective human CYP3A4 inhibitor. A mutilin derivative |
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Azamulin Upstream-Materialien And Downstream Produkte |
Upstream-Materialien
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Downstream Produkte
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Azamulin Anbieter Lieferant Produzent Hersteller Vertrieb Händler. Global( 8)Lieferanten |
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SA 85530b
14-O-(5-(2-Amino1,3,4-triazolyl)thioacetyl)dihydromutilin
76530-44-4
Antibiotic TDM 85-530
Azamulin
All Inhibitors
C24H38N4O4S
Inhibitors
Intermediates & Fine Chemicals
Pharmaceuticals
[(5-Amino-1H-1,2,4-triazol-3-yl)thio]acetic acid (3aS,4R,5S,6R,8R,9R,9aR,10R)-6-ethyldecahydro-5-hydroxy-4,6,9,10-tetramethyl-1-oxo-3a,9-propano-3aH-cyclopentacycloocten-8-yl ester
TMD 85-530, SA 85530b
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