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CAS番号. | 201943-63-7 |
化学名: | |
别名: | |
英語化学名: | LY 341495 |
英語别名: | LY 341495;(2S)-2-AMINO-2-[(1S,2S)-2-CARBOXYCYCLOPROP-1-YL]-3-(XANTH-9-YL) PROPANOIC ACID;(alphaS)-alpha-Amino-alpha-[(1S,2S)-2-carboxycyclopropyl]-9H-xanthene-9-propanoic acid;(alphaS)-alpha-Amino-alpha-[(1S,2S)-2-carboxycyclopropyl]-9H-xanthene-9-propanoic acid LY 341495 |
CBNumber: | CB0200679 |
分子式: | C20H19NO5 |
分子量: | 353.37 |
MOL File: | 201943-63-7.mol |
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LY 341495 化学特性,用途語,生産方法 |
生物活性
Highly potent and selective group II metabotropic glutamate receptor antagonist (K i /IC 50 values are 2.3, 1.3, 173, 990, 6800, 8200 and 22000 nM for human mGlu 2 , mGlu 3 , mGlu 8 , mGlu 7a , mGlu 1a , mGlu 5a and mGlu 4a receptors respectively). Readily brain penetrant and active in vivo . Also available as part of the Group II mGlu Receptor Tocriset™ , Group III mGlu Receptor Tocriset™ and Mixed mGlu Receptor Tocriset™ . |
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LY 341495 上流と下流の製品情報 |
原材料
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準備製品
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LY 341495 生産企業 Global( 18)Suppliers |
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