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3-ethyl-2-(ethylimino)-5-(5-isopropyl-4-methoxy-2-methylbenzylidene)-1,3-thiazolidin-4-one
ethyl 2-(isobutyrylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 4-(3-bromophenyl)-6-(4-methoxyphenyl)-2-oxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate
ethyl 2-{[(4-methylphenyl)sulfanyl]methyl}-3-quinolinecarboxylate
ethyl 2-({[(5,6-dimethyl-4-oxo-3-phenyl-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl)sulfanyl]acetyl}amino)-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
ethyl 6-bromo-2-[(dibenzylamino)methyl]-5-hydroxy-1-methyl-1H-indole-3-carboxylate
2-[(8-ethyl-2-phenyl-4-quinazolinyl)sulfanyl]-N-(1-naphthyl)acetamide
ethyl [6-(4-bromophenyl)-3-methylimidazo[2,1-b][1,3]thiazol-2-yl]acetate
ethyl 4-{2,5-dimethyl-3-[(2,4,6-trioxo-1-phenyltetrahydro-5(2H)-pyrimidinylidene)methyl]-1H-pyrrol-1-yl}benzoate
ethyl3-[({[4-amino-5-(phenoxymethyl)-4H-1,2,4-triazol-3-yl]thio}acetyl)amino]benzoate
ethyl 2-[(5-bromo-2-furoyl)amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
ethyl 7-[4-(benzyloxy)-3-methoxyphenyl]-5-methyl-4,7-dihydrotetraazolo[1,5-a]pyrimidine-6-carboxylate
ethyl 2-({[(5-chloro-3-pyridinyl)oxy]acetyl}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
5-{[1-(2-ethylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylene}-1-phenyl-2,4,6(1H,3H,5H)-pyrimidinetrione
ethyl (6-amino-5-cyano-4-{3-ethoxy-4-[2-(4-morpholinyl)ethoxy]phenyl}-2,4-dihydropyrano[2,3-c]pyrazol-3-yl)acetate
ethyl 1-[4-(3,4-dichlorophenyl)-1,3-thiazol-2-yl]-6,8-difluoro-7-(4-morpholinyl)-4-oxo-1,4-dihydro-3-quinolinecarboxylate
ethyl 2-{[3-(acetyloxy)benzoyl]amino}-2',4-bithiophene-3-carboxylate
ethyl 4-({5-[4-(cyanomethoxy)-3-ethoxybenzylidene]-3-methyl-4-oxo-1,3-thiazolidin-2-ylidene}amino)benzoate
ethyl 3-[2-(4-bromophenyl)-2-oxoethyl]-4-oxo-3,5,6,8-tetrahydropyrido[4',3':4,5]thieno[2,3-d]pyrimidine-7(4H)-carboxylate
4-ethyl-2-({2-[1-(2-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]-2-oxoethyl}sulfanyl)-7,7-dimethyl-5-oxo-5,6,7,8-tetrahydro-3-quinolinecarbonitrile
ethyl {[6-({[(1-benzyl-1H-tetraazol-5-yl)sulfanyl]acetyl}amino)-1,3-benzothiazol-2-yl]sulfanyl}acetate
ethyl 5-amino-1-(4-methylbenzyl)-1H-1,2,3-triazole-4-carboxylate
ethyl 5-amino-1-(3-benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)-1H-pyrazole-4-carboxylate
ethyl 5-[(dimethylamino)carbonyl]-2-[(2-iodobenzoyl)amino]-4-methyl-3-thiophenecarboxylate
2-ethyl-N-(2-{[6-(1H-pyrazol-1-yl)-3-pyridazinyl]amino}ethyl)butanamide
3-ethyl-2-[(3-hydroxyphenyl)imino]-5-(5-methoxy-3-methyl-1,3-benzothiazol-2(3H)-ylidene)-1,3-thiazolidin-4-one
3-(4-ethylphenyl)-2-{[(1-phenyl-1H-tetraazol-5-yl)sulfanyl]methyl}-4(3H)-quinazolinone
2-({1-ethyl-4-nitro-1H-pyrazol-3-yl}carbonyl)-7-{3-nitrobenzylidene}-3-{3-nitrophenyl}-3,3a,4,5,6,7-hexahydro-2H-indazole
ethyl 5-[4-(allyloxy)phenyl]-2-(3-hydroxybenzylidene)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
4-ethyl-N-isopentylbenzamide
ethyl (2-chloro-4-{[3-(4-chlorobenzyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}phenoxy)acetate
ethyl 3-[(2,5-dimethoxyanilino)carbonyl]-2-(2-furoylamino)-4,7-dihydrothieno[2,3-c]pyridine-6(5H)-carboxylate
ethyl 4-{[2-(benzoylamino)-5-ethyl-3-thienyl]methyl}-1-piperazinecarboxylate
ethyl 2-(2-amino-3-cyano-4-(4-ethylphenyl)-7,7-dimethyl-5-oxo-5,6,7,8-tetrahydro-1(4H)-quinolinyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 2-{[(5-{4-nitrobenzylidene}-4-oxo-2-thioxo-1,3-thiazolidin-3-yl)methyl]amino}benzoate
ethyl 3-[(2-methylquinolin-4-yl)amino]benzoate
ethyl 1-(2-chlorobenzyl)-5-{[(4-methyl-1-piperidinyl)acetyl]amino}-1H-1,2,3-triazole-4-carboxylate
ethyl 2-[({4-nitro-1H-pyrazol-1-yl}acetyl)amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
3-(2-ethylphenyl)-2-[(2-ethylphenyl)imino]-5-({6-nitro-1,3-benzodioxol-5-yl}methylene)-1,3-thiazolidin-4-one
ethyl 3-[(2-ethoxyanilino)carbonyl]-2-[(2,4,5-trimethoxybenzyl)amino]-4,7-dihydrothieno[2,3-c]pyridine-6(5H)-carboxylate
ethyl 2-(2,3-dimethoxybenzylidene)-5-(4-fluorophenyl)-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 7-oxo-5,7,9,10-tetrahydro-spiro(6H-benzo[h][1,3]thiazolo[2,3-b]quinazoline-6,1'-cyclopentane)-10-carboxylate
ethyl 2-{[5-(2-{4-nitrophenyl}carbohydrazonoyl)-2-methoxybenzyl]oxy}benzoate
2-({5-[1-(4-ethylphenoxy)ethyl]-4-methyl-4H-1,2,4-triazol-3-yl}sulfanyl)-N-(2-methylphenyl)acetamide
ethyl 4-(4-{4-[(4-ethoxy-4-oxobutanoyl)amino]phenoxy}anilino)-4-oxobutanoate
ethyl2-(2,3-dihydro-1,4-benzodioxin-6-ylmethylene)-5-(2,5-dimethoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 4-{[(2-oxo-1,2-dihydrobenzo[cd]indol-6-yl)sulfonyl]amino}benzoate
ethyl 2-[(4-tert-butylbenzoyl)amino]-5-{3-chloro-4-[(3-fluorobenzyl)oxy]-5-methoxybenzylidene}-4-oxo-4,5-dihydro-3-thiophenecarboxylate
ethyl 5-(3-ethoxy-4-methoxyphenyl)-2-(3-hydroxybenzylidene)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
2-[(6-ethyl-4-methyl-2-oxo-2H-chromen-7-yl)oxy]-N-(4-methylphenyl)acetamide
ethyl 4-({3-[5-(4-chlorobenzylidene)-2,4-dioxo-1,3-thiazolidin-3-yl]propanoyl}amino)benzoate
ethyl 2-amino-1-(4-methoxyphenyl)-7,7-dimethyl-5-oxo-4-(2-thienyl)-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl 5-(4-chlorophenyl)-2-[4-(dimethylamino)benzylidene]-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
3-ethyl-5-[2-(3-ethyl-6-methoxy-1,3-benzothiazol-2(3H)-ylidene)-1-phenylethylidene]-2-[(4-methylphenyl)imino]-1,3-thiazolidin-4-one
ethyl 2-{[(1,3-benzothiazol-2-ylsulfanyl)acetyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 5-{[(4-fluoro-2-methylphenyl)sulfonyl]amino}-2-methyl-1-benzofuran-3-carboxylate
ethyl 2-{[2-(3-benzoylphenyl)propanoyl]amino}benzoate
ethyl 2-[(2-methoxybenzoyl)amino]-4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-3-carboxylate
2-({1-ethyl-4-nitro-1H-pyrazol-3-yl}carbonyl)-7-{4-nitrobenzylidene}-3-{4-nitrophenyl}-3,3a,4,5,6,7-hexahydro-2H-indazole
ethyl 3-(2-hydroxyethyl)-2-[(4-methoxyphenyl)imino]-4-methyl-2,3-dihydro-1,3-thiazole-5-carboxylate
3-ethyl-5-[2-(3-ethyl-6-methoxy-1,3-benzothiazol-2(3H)-ylidene)-1-phenylethylidene]-2-thioxo-1,3-thiazolidin-4-one
ethyl 5-(aminocarbonyl)-2-({3-nitro-4-methoxybenzoyl}amino)-4-methyl-3-thiophenecarboxylate
ethyl 5-(2,5-dimethoxyphenyl)-7-methyl-2-[(6-methyl-1,3-benzodioxol-5-yl)methylene]-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-methyl-4-(1-naphthyl)-5-oxo-4,5-dihydro-1H-indeno[1,2-b]pyridine-3-carboxylate
ethyl 5-(3-methoxyphenyl)-7-methyl-3-oxo-2-{[5-(1-piperidinyl)-2-furyl]methylene}-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl {[8-(4-methoxyphenyl)-7-oxo-5,6,7,8-tetrahydronaphtho[2',1':4,5]thieno[2,3-d]pyrimidin-9-yl]sulfanyl}acetate
1-ethyl-4-[3-(4-isopropylphenyl)acryloyl]piperazine
ethyl 4-[2-(aminocarbonyl)anilino]-4-oxobutanoate
4-(4-ethylphenyl)-N-(4-fluorophenyl)-2-methyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxamide
ethyl 3-({[1-(4-methylphenyl)-1H-1,2,4-triazol-3-yl]carbonyl}amino)benzoate
ethyl 6-{[2-(4-chlorophenyl)-2-oxoethyl]sulfanyl}-5-cyano-4-isobutyl-2-methyl-1,4-dihydro-3-pyridinecarboxylate
ethyl 2-amino-4-(3-iodophenyl)-5-oxo-4H,5H-pyrano[2,3-b]chromene-3-carboxylate
ethyl 2-[({[3-cyano-6-methyl-4-(2-thienyl)-5,6,7,8-tetrahydro[1,6]naphthyridin-2-yl]sulfanyl}acetyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 5-oxo-1-phenyl-6-(3-pyridinylmethyl)-1,5-dihydro[1,2,4]triazolo[3,4-c][1,2,4]triazine-3-carboxylate
ethyl 2-({[2-(4-ethylphenyl)-4-quinolinyl]carbonyl}amino)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 1-(4-chlorophenyl)-5-ethoxy-2-methyl-1H-indole-3-carboxylate
ethyl 2-(3,4-dichlorobenzylidene)-5-{3-nitrophenyl}-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
1-({1-ethyl-4-nitro-1H-pyrazol-3-yl}carbonyl)piperidine
ethyl 1-(4-chlorophenyl)-8-oxo-9-phenyl-4,6-dithia-1,2,9-triazaspiro[4.4]non-2-ene-3-carboxylate
ethyl 5-(4-methoxyphenyl)-7-methyl-2-{[5-(4-morpholinyl)-2-furyl]methylene}-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
2-({5-[1-(4-ethylphenoxy)ethyl]-4-methyl-4H-1,2,4-triazol-3-yl}sulfanyl)-N-(4-phenyl-1,3-thiazol-2-yl)acetamide
ethyl {[10-(4-methoxyphenyl)-2-methyl-8,9-dihydro-7H-cyclopenta[5',6']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-yl]sulfanyl}acetate
ethyl 4-({[(4-ethyl-5-{[(4-methoxybenzoyl)amino]methyl}-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}amino)benzoate
ethyl 7-(methylsulfanyl)-4,5-dihydro-3H-1-thia-3,5,6,8-tetraazaacenaphthylene-2-carboxylate
ethyl 2-amino-4-(2-chlorophenyl)-6-(hydroxymethyl)-8-oxo-4,8-dihydropyrano[3,2-b]pyran-3-carboxylate
5-(4-ethylphenyl)-1H-pyrazole-3-carbaldehyde
ethyl {2-[chloro(difluoro)methyl]-5-formyl-1,3-benzodioxol-2-yl}acetate
ethyl 5-(4-fluorophenyl)-2-[(3-methyl-2-thienyl)methylene]-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 4-(4-iodophenyl)-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate
ethyl 2-{3-[(4-iodophenoxy)methyl]-4-methoxybenzylidene}-5-(4-methoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 5-(1,3-benzodioxol-5-yl)-2-(2-methoxybenzylidene)-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 7-chloro-4-phenyl-2-(trifluoromethyl)-2H-pyrido[1,2-a][1,3,5]triazine-2-carboxylate
ethyl 5-(4-chlorophenyl)-2-(4-hydroxy-3-methoxybenzylidene)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-[(tetrahydro-2-furanylcarbonyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
1-ethyl-9-hydroxy-2,5,7-trimethyl-1H-imidazo[4',5':5,6]pyrido[2,3-d]pyrimidine-6,8(5H,7H)-dione
ethyl 5-(3-chloro-4-methylphenyl)-4,6-dioxo-1,3a,4,5,6,6a-hexahydropyrrolo[3,4-c]pyrazole-3-carboxylate
ethyl 2-{[(3,4-dimethoxyphenyl)acetyl]amino}-4,5-dimethyl-3-thiophenecarboxylate
ethyl 3-[(2-methyl-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl)oxy]benzoate
ethyl 2-[5-(3-chloro-4-hydroxy-5-methoxybenzylidene)-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate
ethyl 4-[(2,6-dimethylanilino)sulfonyl]benzylcarbamate
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