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ethyl 2-amino-5-[(diethylamino)carbonyl]-4-methyl-3-thiophenecarboxylate
ethyl 4-(abieta-8,11,13-trien-18-ylamino)-2-(methylsulfanyl)-5-pyrimidinecarboxylate
ethyl 2-[5-nitro-2-(1-pyrrolidinyl)benzylidene]-5-(2-methoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 11-(4-chlorophenyl)-7-(2-thienyl)-5,6,7,11-tetrahydrobenzo[h][1,2,4]triazolo[3,4-b]quinazoline-9-carboxylate
ethyl 2-[({[(4-chloro-1,3-dimethyl-1H-pyrazol-5-yl)carbonyl]amino}carbothioyl)amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
ethyl 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-{3-nitrophenyl}-1H-1,2,3-triazole-4-carboxylate
ethyl 4-{[3-cyano-6-(2-thienyl)-4-(3-thienyl)-2-pyridinyl]sulfanyl}-3-oxobutanoate
4-ethyl 2-methyl 3-methyl-5-({[(2-methyl-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl)sulfanyl]acetyl}amino)-2,4-thiophenedicarboxylate
ethyl 4-({cyclohexyl[(4-fluorophenyl)sulfonyl]amino}acetyl)piperazine-1-carboxylate
6-ethyl 8-methyl 5-amino-3-oxo-7-(3-pyridinyl)-2-(3-pyridinylmethylene)-2,3-dihydro-7H-[1,3]thiazolo[3,2-a]pyridine-6,8-dicarboxylate
ethyl 5-hydroxynicotinate
3-ethyl-5-(3-ethyl-1,3-benzothiazol-2(3H)-ylidene)-2-[(4-hydroxyphenyl)imino]-1,3-thiazolidin-4-one
2-[(4-{[(3-ethyl-5-sulfanyl-4H-1,2,4-triazol-4-yl)imino]methyl}-2-methoxyphenoxy)methyl]benzonitrile
ethyl 5-({[2-(acetylamino)-3-(1H-indol-3-yl)propanoyl]amino}methyl)-2-furoate
ethyl 2-bromo-3-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)propanoate
ethyl 2-[(2,5-dichlorobenzoyl)amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
ethyl 4-[(2-furylmethyl)amino]-8-(trifluoromethyl)-3-quinolinecarboxylate
ethyl 4-(4-bromophenyl)-5-cyano-2-methyl-6-[(2-thienylmethyl)sulfanyl]-1,4-dihydro-3-pyridinecarboxylate
ethyl 2-[(3-methoxy-2-naphthoyl)amino]-4,5-dimethyl-3-thiophenecarboxylate
ethyl 2-{[1-(cyanomethyl)-1H-indol-3-yl]methylene}-5-(3-methoxyphenyl)-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 4-cyano-3-methyl-5-{[3-(1-methyl-1H-pyrazol-4-yl)acryloyl]amino}-2-thiophenecarboxylate
ethyl 5-(2,7-dimethoxy-1-naphthyl)-7-methyl-3-oxo-2-(3-pyridinylmethylene)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
3-[2-(4-ethylphenyl)-2-oxoethyl]-3-hydroxy-1,3-dihydro-2H-indol-2-one
2-(4-ethylphenoxy)-N-[4-(4-{[(4-ethylphenoxy)acetyl]amino}benzyl)phenyl]acetamide
ethyl 2-(2-hydroxy-3-methoxybenzylidene)-7-methyl-3-oxo-5-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 3-amino-6-phenyl-4-(2-thienyl)furo[2,3-b]pyridine-2-carboxylate
ethyl 2-{3-ethoxy-4-[(4-fluorobenzyl)oxy]benzylidene}-7-methyl-3-oxo-5-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl {2-bromo-6-ethoxy-4-[(2-methyl-5-oxo-1,3-oxazol-4(5H)-ylidene)methyl]phenoxy}acetate
ethyl 2-(butyrylamino)-4,5,6,7,8,9,10,11,12,13-decahydrocyclododeca[b]thiophene-3-carboxylate
5-[2-(1-ethyl-3,3-dimethyl-5-phenyl-1,3-dihydro-2H-indol-2-ylidene)ethylidene]-3-phenyl-2-thioxo-1,3-thiazolidin-4-one
ethyl 2-(4-isopropylbenzylidene)-5-(2-methoxy-1-naphthyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-({[2-(5-ethyl-2-thienyl)-4-quinolinyl]carbonyl}amino)-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
2-ethyl-N-(5-methyl-4-phenyl-1,3-thiazol-2-yl)hexanamide
ethyl 6-bromo-5-hydroxy-1-methyl-2-(1-piperidinylmethyl)-1H-indole-3-carboxylate
4-{3-[(3-ethyl-2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-dimethyl-1H-pyrrol-1-yl}benzenesulfonamide
ethyl 2-[({2-nitrophenyl}sulfanyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 5-(4-methoxyphenyl)-3-{[(4-methyl-1-piperazinyl)carbothioyl]amino}-2-thiophenecarboxylate
ethyl 4-({[4-oxo-2-(4-toluidino)-5,6-dihydro-4H-1,3-thiazin-6-yl]carbonyl}amino)benzoate
ethyl 2-({[6-bromo-2-(4-butylphenyl)-4-quinolinyl]carbonyl}amino)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 3-allyl-8-(benzoylamino)-3,4-dihydro-2H-thieno[3,2-h][1,3]benzoxazine-7-carboxylate
ethyl 6-(5-bromo-2-methoxyphenyl)-8-methyl-4-oxo-3,4-dihydro-2H,6H-pyrimido[2,1-b][1,3]thiazine-7-carboxylate
ethyl 4-{3-[(4-chlorophenoxy)methyl]-4-methoxyphenyl}-2-methyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl 3-methoxy-4-{[(4-methylphenyl)sulfonyl]oxy}benzoate
ethyl 5-(4-bromophenyl)-2-[(6-chloro-1,3-benzodioxol-5-yl)methylene]-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 4-[(5-{[2,5-dimethyl-1-(3-pyridinyl)-1H-pyrrol-3-yl]methylene}-3-methyl-4-oxo-1,3-thiazolidin-2-ylidene)amino]benzoate
ethyl 4-(1,5-dimethyl-1H-pyrazol-4-yl)-2-methyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl 2-({[(3-allyl-7-methyl-4-oxo-3,4,5,6,7,8-hexahydro[1]benzothieno[2,3-d]pyrimidin-2-yl)sulfanyl]acetyl}amino)-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
2-(ethyloxy)ethyl 2,7,7-trimethyl-4-(4-methylphenyl)-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate
ethyl 3-(2-amino-3,4-dioxo-1-cyclobuten-1-yl)acrylate
ethyl cyano[(4-{[(4,6-dimethyl-2-pyrimidinyl)amino]sulfonyl}phenyl)hydrazono]acetate
ethyl 2-[(1,5-dimethyl-1H-pyrazol-4-yl)methylene]-5-(4-fluorophenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 4-(2-thienyl)-4,5-dihydro-1H-pyrazole-3-carboxylate
ethyl 5-methyl-2-[(4-methyl-1-piperazinyl)sulfonyl]phenyl ether
3-(4-ethylphenyl)-2-(4-fluorophenyl)-1,3-thiazolidin-4-one
ethyl 2-{[3-(difluoromethoxy)benzoyl]amino}-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
ethyl 2-(5,6-dichloro-1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-4-methylpentanoate
ethyl 2-amino-4-(2-fluorophenyl)-7-methyl-5-oxo-4H,5H-pyrano[4,3-b]pyran-3-carboxylate
ethyl 4-[(2-ethyl-4-methyl-1H-imidazol-1-yl)sulfonyl]-1-naphthyl ether
ethyl 4-(4-fluorophenyl)-2-({[(2-methyl-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl)sulfanyl]acetyl}amino)-3-thiophenecarboxylate
ethyl 2-{[(4-bromo-3-methylphenoxy)acetyl]amino}-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
ethyl2-{[(6-{[2-(ethoxycarbonyl)anilino]carbonyl}-2-pyridinyl)carbonyl]amino}benzoate
ethyl 4-(acetyloxy)-5-({2-nitrophenyl}sulfanyl)-2-methyl-3-thiophenecarboxylate
ethyl 2-methyl-4-[(2-methyl-2,3-dihydro-1H-indol-1-yl)sulfonyl]phenyl ether
ethyl (6-bromo-4-phenyl-2-(3,4,5-trimethoxyphenyl)-3(4H)-quinazolinyl)acetate
ethyl 6-methyl-2-[(2-methylbenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 4-{5-[2-(cyanoacetyl)carbohydrazonoyl]-2-furyl}benzoate
ethyl 4-[(2-phenylbutanoyl)amino]benzoate
1-ethyl-5-methyl-N-(4-pyridinyl)-1H-pyrazole-4-carboxamide
ethyl 2-({5-chloro-2-nitrobenzoyl}amino)-1-benzothiophene-3-carboxylate
ethyl 2-amino-5-oxo-1-phenyl-4-(3-pyridinyl)-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl 2-[(diethoxyphosphorothioyl)sulfanyl]-3-[4-({2-[(diethoxyphosphorothioyl)sulfanyl]-3-ethoxy-1-methyl-3-oxo-1-propenyl}amino)anilino]-2-butenoate
ethyl2-{3-ethoxy-4-[(4-fluorobenzyl)oxy]benzylidene}-5-(4-methoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
5-ethyl-2-methylphenyl 4-fluorobenzoate
ethyl 5,5-dimethyl-2-{[4-(1-piperidinyl)butanoyl]amino}-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylate
ethyl 2-({3-[(2-fluoroanilino)carbonyl]-2H-chromen-2-ylidene}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 5-(2-methoxybenzylidene)-2-methyl-4-oxo-4,5-dihydro-1H-pyrrole-3-carboxylate
ethyl 2-{[(acetyloxy)(phenyl)acetyl]amino}-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 5-[(diethylamino)carbonyl]-2-(2-furoylamino)-4-methyl-3-thiophenecarboxylate
ethyl 4-(1-benzyl-4(1H)-pyridinylidene)-2-cyano-2-butenoate
ethyl 2-({[1-(4-chlorophenyl)-5-oxo-3-pyrrolidinyl]carbonyl}amino)benzoate
ethyl 2-{[5-(2-cyanophenyl)-2-furyl]methylene}-5-[4-(dimethylamino)phenyl]-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 1,2-dimethyl-4-{[(methylamino)carbothioyl]amino}-1H-imidazole-5-carboxylate
ethyl 6,7-dichloro-4-hydroxy-3-quinolinecarboxylate
ethyl 4-[4-(2-amino-2-oxoethoxy)phenyl]-6-methyl-2-thioxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate
ethyl 7-methyl-2-[(1-methyl-1H-pyrazol-4-yl)methylene]-3-oxo-5-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 5-[(3,4-dimethylbenzoyl)amino]-2-hydroxybenzoate
ethyl 4-{3-methoxy-4-[(4-methoxyphenoxy)methyl]phenyl}-2-methyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl 2-[({[(benzoylsulfanyl)acetyl]oxy}acetyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 4-{[(1,3-diethyl-2,4,6-trioxotetrahydro-5(2H)-pyrimidinylidene)methyl]amino}benzoate
1-[4-(ethyloxy)phenyl]-3-[(4-methylphenyl)amino]pyrrolidine-2,5-dione
ethyl 2-anilino-5-(3-hydroxy-4-methoxybenzylidene)-4-oxo-4,5-dihydro-3-thiophenecarboxylate
ethyl 4-acetyl-1-(4-ethoxyphenyl)-5-methyl-1H-pyrazole-3-carboxylate
3-(4-ethylphenyl)-2-{[2-(4-morpholinyl)-2-oxoethyl]sulfanyl}-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3H)-one
ethyl 2-(1-benzoyl-2,2,6,7-tetramethyl-3-thioxo-2,3-dihydro-4(1H)-quinolinylidene)-5-phenyl-1,3-dithiole-4-carboxylate
ethyl 4-{[(2-phenylcyclopropyl)carbonyl]amino}benzoate
3-ethyl-2-[(2-ethylphenyl)imino]-5-[(2-propoxy-1-naphthyl)methylene]-1,3-thiazolidin-4-one
ethyl 1-(3-chlorophenyl)-5,7-diphenyl-1,5-dihydro[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxylate
ethyl 3-amino-6,6-dimethyl-5,6,7,8-tetrahydrothieno[2,3-b]quinoline-2-carboxylate
ethyl 5-(4-isopropoxyphenyl)-7-methyl-2-[(3-methyl-2-thienyl)methylene]-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-[(5-{2-chloro-5-nitrophenyl}-2-furyl)methylene]-5-[4-(dimethylamino)phenyl]-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
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