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ethyl 5-(2-chlorophenyl)-2-[(2-isopropoxy-1-naphthyl)methylene]-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
3-{[1-(4-ethylphenyl)-3,5-dioxo-4-pyrazolidinylidene]methyl}phenyl acetate
ethyl 4-(4-methoxyphenyl)-5-methyl-2-[(2-thienylcarbonyl)amino]-3-thiophenecarboxylate
ethyl 1-(4-ethoxyphenyl)-6-methyl-5-oxo-1,5-dihydro[1,2,4]triazolo[3,4-c][1,2,4]triazine-3-carboxylate
1-ethyl-3-hydroxy-3-{2-oxo-2-[4-(1H-pyrrol-1-yl)phenyl]ethyl}-1,3-dihydro-2H-indol-2-one
ethyl 2-amino-1-(4-bromophenyl)-5-oxo-4-(2-thienyl)-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl 4-(4-bromophenyl)-2-{[(2-methylphenoxy)acetyl]amino}-3-thiophenecarboxylate
5-ethyl-2-(2-toluidino)-1,3-thiazol-4(5H)-one
ethyl 5-(4-chlorophenyl)-2-(2-methoxybenzylidene)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-(4-bromophenyl)-4-quinolinecarboxylate
ethyl 4-(1,3-benzodioxol-5-yl)-7-(4-chlorophenyl)-2-methyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl phenyl(2H-1,2,3-triazol-4-ylsulfanyl)acetate
ethyl 1-[1-(3-methylphenyl)-2,5-dioxo-3-pyrrolidinyl]-3-piperidinecarboxylate
ethyl 4-(1,5-dimethyl-1H-pyrazol-4-yl)-6-methyl-2-thioxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate
ethyl 2-[methacryloyl(methyl)amino]benzoate
ethyl 2-amino-5-cyano-6-methyl-4-[2-(trifluoromethyl)phenyl]-4H-pyran-3-carboxylate
ethyl 2-[4-(difluoromethoxy)benzylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 5-(6-bromo-1,3-dioxo-1H-benzo[de]isoquinolin-2(3H)-yl)-2-chlorobenzoate
ethyl 6,8-dimethylthieno[2,3-b]quinoline-2-carboxylate
ethyl 2-(3-bromo-4-ethoxybenzylidene)-5-(4-ethoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 6-methyl-4-(5-methyl-2-furyl)-2-oxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate
ethyl {[5-(2-bromophenyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetate
ethyl 4-{3-(2-thienyl)-2-[(2-thienylcarbonyl)amino]acryloyl}-1-piperazinecarboxylate
3-ethyl-6-(3,4,5-trimethoxyphenyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
5-ethyl-2-methoxy-N-[2-(5-methoxy-2-methyl-1H-indol-3-yl)ethyl]benzenesulfonamide
ethyl 2-[(2-thienylcarbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 2-(benzoylamino)-4-methyl-5-(4-toluidinocarbonyl)-3-thiophenecarboxylate
ethyl 6-chloro-4-[(3-pyridinylmethyl)amino]-3-quinolinecarboxylate
ethyl 6-methyl-2-{[(4-methyl-1,4-diazepan-1-yl)carbothioyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 4-methyl-2-[(2-methyl-3-furoyl)amino]-1,3-thiazole-5-carboxylate
ethyl 5-(4-isopropylphenyl)-7-methyl-2-{[5-(4-methyl-1-piperazinyl)-2-furyl]methylene}-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 3-amino-2-[(cyanomethyl)sulfanyl]-4-oxo-3,5,6,8-tetrahydropyrido[4',3':4,5]thieno[2,3-d]pyrimidine-7(4H)-carboxylate
ethyl [(3-allyl-4-oxo-3,5,6,7,8,9-hexahydro-4H-cyclohepta[4,5]thieno[2,3-d]pyrimidin-2-yl)sulfanyl]acetate
ethyl 2-amino-7,7-dimethyl-5-oxo-4-phenyl-5,6,7,8-tetrahydro-4H-chromene-3-carboxylate
ethyl 2-(2,4-dichlorobenzylidene)-5-(2-fluorophenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 6-ethyl-2-{[(5-methyl-3-phenyl-4-isoxazolyl)carbonyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 2,5-bis(4-methoxyphenyl)-1,3-dioxolane-4-carboxylate
ethyl 3-(4-imidazo[1,2-a]pyridin-2-ylphenyl)acrylate
ethyl 4-[2-{[4-(ethoxycarbonyl)phenyl]imino}-5-(3-hydroxybenzylidene)-4-oxo-1,3-thiazolidin-3-yl]benzoate
ethyl 10-(3-chloropropanoyl)-5-oxido-10H-phenothiazin-2-ylcarbamate
2-(ethyloxy)ethyl 4-[3,4-bis(methyloxy)phenyl]-2-methyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate
ethyl 4-{5-[7-butyryl-3-(methylsulfanyl)-6,7-dihydro[1,2,4]triazino[5,6-d][3,1]benzoxazepin-6-yl]-2-furyl}benzoate
ethyl 2-[3-benzoyl-2-(3-chlorophenyl)-4-hydroxy-5-oxo-2,5-dihydro-1H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
ethyl 2-{[(2-bromo-4-methylphenoxy)acetyl]amino}-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
2-[(7-ethyl-1,3-dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)sulfanyl]-N-(3-fluorophenyl)acetamide
ethyl 2,3-dihydro-1H-inden-5-ylcarbamate
ethyl 3-[3-(3-pyridinyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]phenyl ether
ethyl 2-{[(4-isopropyl-3-methylphenoxy)acetyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl (2-{2-[(2-bromo-4-methylphenoxy)acetyl]carbohydrazonoyl}phenoxy)acetate
ethyl 4-{[4-fluoro(phenylsulfonyl)anilino]acetyl}-1-piperazinecarboxylate
ethyl 1-(2-chloro-6-fluorobenzyl)-3-methyl-1H-pyrazole-5-carboxylate
ethyl bromo(cyclohexyl)acetate
4'-(5-ethyl-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl hexyl ether
ethyl 2-{[(4-bromo-2-methylphenoxy)acetyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 2-(3-chloro-4-ethoxybenzylidene)-5-(2,5-dimethoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
5-{5-[(1-(4-ethylphenyl)-4,6-dioxo-2-thioxotetrahydro-5(2H)-pyrimidinylidene)methyl]-2-furyl}-2-methylbenzoic acid
2-{[4-ethyl-5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-phenylacetamide
5-ethyl-N-(4-methylphenyl)-1-(2-pyridinyl)-1H-pyrazole-4-carboxamide
4-ethyl 2-methyl 5-{[(acetyloxy)(phenyl)acetyl]amino}-3-methyl-2,4-thiophenedicarboxylate
ethyl 5-(4-chlorophenyl)-2-methyl-1-{[(2-methyl-1H-benzimidazol-1-yl)acetyl]amino}-1H-pyrrole-3-carboxylate
ethyl 4-({3-[(3-allyl-5,6-dimethyl-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl)sulfanyl]propanoyl}amino)benzoate
ethyl 2-({[(cyclobutylcarbonyl)amino]carbothioyl}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 2-{[(4-chloro-2-methylphenoxy)acetyl]amino}-6-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
3-ethyl-2-[3-(3-ethyl-1,3-thiazolidin-2-ylidene)-1-propenyl]-4,5-dihydro-1,3-thiazol-3-ium
ethyl 2-{[5-(diethylamino)-2-furyl]methylene}-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 3-chloro-4-methyl-1-benzothiophene-2-carboxylate
ethyl 5-ethyl-2-{[(4-oxo-3(4H)-quinazolinyl)acetyl]amino}-3-thiophenecarboxylate
ethyl 7-amino-3-[(2-fluorophenyl)diazenyl]-2-oxo-1,2-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate
ethyl 2-amino-4-(2,3-dichlorophenyl)-6-(hydroxymethyl)-8-oxo-4,8-dihydropyrano[3,2-b]pyran-3-carboxylate
ethyl 2-[(4-methoxybenzoyl)amino]-5-methyl-4-phenylthiophene-3-carboxylate
ethyl 3-[(3-ethoxybenzoyl)amino]-4-(4-morpholinyl)benzoate
ethyl 5-({5-benzyl-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}sulfanyl)[1,2,3]triazolo[1,5-a]quinazoline-3-carboxylate
ethyl 2-[4-(acetyloxy)-3-ethoxybenzylidene]-5-[4-(allyloxy)-3-ethoxyphenyl]-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 5-(2,5-dimethoxybenzylidene)-2-methyl-4-oxo-4,5-dihydro-1H-pyrrole-3-carboxylate
ethyl [2-chloro-4-({2-[(4-methoxyphenyl)imino]-3-methyl-4-oxo-1,3-thiazolidin-5-ylidene}methyl)phenoxy]acetate
ethyl 4-(3,4-dimethylphenyl)-2-[(3-methylbutanoyl)amino]-3-thiophenecarboxylate
ethyl 6-amino-5-cyano-2-propyl-4-(4-pyridinyl)-4H-pyran-3-carboxylate
ethyl 6-tert-butyl-2-[(3-{4-nitrophenyl}acryloyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 4-amino-2-{[2-(4-methoxyanilino)-2-oxoethyl]sulfanyl}-5-pyrimidinecarboxylate
6-ethyl-2-[(2,3,4,5,6-pentafluorobenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
5'-ethyl 3'-(2-methoxyethyl) 2'-amino-1,3-dihydro-6'-propyl-2-oxospiro[2H-indole-3,4'-(4'H)-pyran]-3',5'-dicarboxylate
ethyl 2-[(4-chlorobenzoyl)amino]-5-[(2-fluoroanilino)carbonyl]-4-methyl-3-thiophenecarboxylate
ethyl 2-{[(2,4-dichlorophenoxy)acetyl]amino}-5-ethyl-3-thiophenecarboxylate
2-[(3-ethyl-4-oxo-3,4-dihydroquinazolin-2-yl)sulfanyl]-N-(3-methylphenyl)acetamide
ethyl 2-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methylene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 5-bromo-2-[2-(4-methoxybenzylidene)hydrazino]-1,3-thiazole-4-carboxylate
ethyl 5-(4-ethoxyphenyl)-7-methyl-3-oxo-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-[(4-methylbenzoyl)amino]-5-phenylthiophene-3-carboxylate
4-ethyl-5-methyl-2-[(phenoxyacetyl)amino]-3-thiophenecarboxamide
5-(5-ethyl-2-thienyl)-N-(3-phenylpropyl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
ethyl 2-{4-[ethyl(methoxycarbonyl)amino]phenyl}-3,3,3-trifluoro-2-hydroxypropanoate
ethyl 2-(3-bromobenzylidene)-7-methyl-5-(4-methylphenyl)-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
3-ethyl-5-[2-(3-ethylnaphtho[2,1-d][1,3]thiazol-2(3H)-ylidene)ethylidene]-2-{[4-(2-phenylvinyl)phenyl]imino}-1,3-thiazolidin-4-one
ethyl (2-{[1-(4-fluorophenyl)-3,5-dioxo-4-pyrazolidinylidene]methyl}phenoxy)acetate
ethyl 5-(2,3-dimethoxyphenyl)-3-oxo-7-phenyl-2-(3,4,5-trimethoxybenzylidene)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-[(2-{[1-(ethoxycarbonyl)-2-oxopropyl]sulfanyl}-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanyl]-3-oxobutanoate
ethyl 2-[(4-fluorobenzoyl)amino]-4-(4-fluorophenyl)-5-methylthiophene-3-carboxylate
ethyl 2-[(4-chlorobenzoyl)amino]-4-ethyl-5-methyl-3-thiophenecarboxylate
ethyl 5-[(diethylamino)carbonyl]-2-[(3,4-dimethoxybenzoyl)amino]-4-methyl-3-thiophenecarboxylate
ethyl 5-(4-chlorophenyl)-2-{[5-(2,4-dichlorophenyl)-2-furyl]methylene}-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
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