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ethyl 2-(2-bromo-4-hydroxy-5-methoxybenzylidene)-7-methyl-3-oxo-5-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-({[5-(5-chloro-2-thienyl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]carbonyl}amino)-5-phenyl-3-thiophenecarboxylate
ethyl 1-[(4-fluoroanilino)carbonyl]-4-piperidinecarboxylate
ethyl 2-(2,5-dimethyl-1H-pyrrol-1-yl)-4-(4-methoxyphenyl)-3-thiophenecarboxylate
ethyl 5-(2-ethoxy-3-methoxyphenyl)-2-(4-isobutoxybenzylidene)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 4-(1,8-dimethyl-16,18-dioxo-17-azapentacyclo[6.6.5.0~2,7~.0~9,14~.0~15,19~]nonadeca-2,4,6,9,11,13-hexaen-17-yl)benzoate
ethyl 5-(4-chlorophenyl)-2-(3,5-diiodo-4-methoxybenzylidene)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 1-benzyl-4-(2-chloro-4-hydroxy-3-iodo-5-methoxyphenyl)-6-methyl-2-oxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate
ethyl 5-(1,3-benzodioxol-5-yl)-2-{[5-(dimethylamino)-2-furyl]methylene}-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 4-methyl-5-{[3-(trifluoromethyl)anilino]carbonyl}-2-[(3,4,5-trimethoxybenzoyl)amino]-3-thiophenecarboxylate
ethyl chloro[(3-methylphenyl)hydrazono]acetate
ethyl [6-amino-4-(4-tert-butylphenyl)-5-cyano-2,4-dihydropyrano[2,3-c]pyrazol-3-yl]acetate
ethyl 2-(3-bromo-4-hydroxy-5-methoxybenzylidene)-5-(3-methoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
2-ethyl-N-(2-ethyl-6-methylphenyl)butanamide
4-ethylphenyl (4-methylphenoxy)acetate
ethyl 2-(1-butyryl-2,2-dimethyl-3-thioxo-2,3-dihydro-4(1H)-quinolinylidene)-5-phenyl-1,3-dithiole-4-carboxylate
ethyl 4-methyl-2-[(3-pyridinylcarbonyl)amino]-5-(4-toluidinocarbonyl)-3-thiophenecarboxylate
ethyl ,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 3-(4-aminophenyl)-2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)propanoate
ethyl 2-{[(4-bromophenyl)sulfonyl]amino}-4-ethyl-5-methyl-3-thiophenecarboxylate
5-ethyl-4-hydroxy-3-(N-hydroxyethanimidoyl)-1,6-diphenyl-2(1H)-pyridinone
ethyl 2-(2-chlorobenzylidene)-7-methyl-3-oxo-5-(2-phenylvinyl)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
2-({1-ethyl-4-nitro-1H-pyrazol-3-yl}carbonyl)-5-methyl-3-(2-thienyl)-7-(2-thienylmethylene)-3,3a,4,5,6,7-hexahydro-2H-indazole
ethyl 2-({1-[4-(ethoxycarbonyl)phenyl]-2,5-dimethyl-1H-pyrrol-3-yl}methylene)-5-(4-methoxy-1-naphthyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 3-(butyrylamino)benzoate
ethyl 2-(2-chlorobenzylidene)-3-oxo-7-phenyl-5-(2-thienyl)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 7-(difluoromethyl)-5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate
ethyl 4-({3-nitro-4-methoxybenzoyl}amino)benzoate
3-ethyl-2-(isopropylsulfanyl)-5,6-dihydrospiro(benzo[h]quinazoline-5,1'-cyclopentane)-4(3H)-one
ethyl 5-(4-fluorophenyl)-2-[3-(1-naphthylmethoxy)benzylidene]-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 3-{[(3-fluorobenzyl)amino]carbonyl}-1-methyl-1H-pyrazole-5-carboxylate
ethyl 3-cyano-6-propyl-4,5,6,7-tetrahydro-1-benzothien-2-ylcarbamate
ethyl 3-[3-(3-methylphenyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]phenyl ether
ethyl 5-{[4-(2-quinoxalinyl)phenoxy]methyl}-2-furoate
ethyl 2-(acetylamino)-7-[(benzoyloxy)imino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 4-{[5-(2-hydroxybenzylidene)-3-methyl-4-oxo-1,3-thiazolidin-2-ylidene]amino}benzoate
ethyl 2-[(2-thienylcarbonyl)amino]-2',4-bithiophene-3-carboxylate
ethyl 2-{[3-(1-methyl-1H-pyrazol-4-yl)acryloyl]amino}-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
ethyl 7-methyl-4-oxo-2-thioxo-5-[2-(trifluoromethyl)phenyl]-1,2,3,4,5,8-hexahydropyrido[2,3-d]pyrimidine-6-carboxylate
2-[(3-ethyl-5,6-dimethyl-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl)sulfanyl]-N-[4-(ethyloxy)phenyl]acetamide
ethyl 2-(4-hydroxy-3-iodo-5-methoxybenzylidene)-7-methyl-3-oxo-5-(2-thienyl)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 4-{[(3,4-diethoxyphenyl)acetyl]amino}benzoate
ethyl 4-amino-2-{[1-methyl-2-oxo-2-(phenylamino)ethyl]sulfanyl}pyrimidine-5-carboxylate
4-ethyl-N-[5-(3-ethyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)-2-methylphenyl]benzamide
ethyl {2-bromo-6-methoxy-4-[2-(4-methylphenyl)carbohydrazonoyl]phenoxy}acetate
ethyl 4-[(4-butoxy-3-methylphenyl)sulfonyl]-1-piperazinecarboxylate
6-ethyl-N-(4-methylphenyl)-2-phenyl-4-quinolinecarboxamide
ethyl 2-({[(3-methylbutanoyl)amino]carbothioyl}amino)-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
ethyl 2-({[3-amino-4-(4-methoxyphenyl)-6-phenylthieno[2,3-b]pyridin-2-yl]carbonyl}amino)-4,5-dimethyl-3-thiophenecarboxylate
ethyl 2-{[(2-chloro-3-pyridinyl)carbonyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 2-[({[(4-bromo-1-ethyl-1H-pyrazol-3-yl)carbonyl]amino}carbothioyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 5-({[1-(4-bromophenyl)-3-methyl-5-oxo-1,5-dihydro-4H-pyrazol-4-ylidene]methyl}amino)-4-cyano-3-methyl-2-thiophenecarboxylate
2-ethyl-7-(1-piperazinyl)-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
2-(4-ethylphenyl)-2-oxoethyl 2-(4-ethoxyphenyl)-4-quinolinecarboxylate
ethyl 3-cyano-2-[({[5-(2-furyl)-1,3,4-oxadiazol-2-yl]sulfanyl}acetyl)amino]-4,7-dihydrothieno[2,3-c]pyridine-6(5H)-carboxylate
ethyl 4-(4-bromophenyl)-2-[(4-fluorobenzoyl)amino]-3-thiophenecarboxylate
2-({4-ethyl-5-[(4-methylphenoxy)methyl]-4H-1,2,4-triazol-3-yl}sulfanyl)-N-[3-(methylsulfanyl)phenyl]acetamide
ethyl 5-{[(4,6-dioxo-1,4,5,6-tetrahydro-2-pyrimidinyl)sulfanyl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
ethyl 2-{[(4-chloro-2-methylphenoxy)acetyl]amino}-4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-3-carboxylate
(2-ethyl-1-methyl-1H-imidazol-5-yl)(2-methoxyphenyl)methanol
ethyl 4-({2-[(5-bromo-2-furoyl)amino]-3-phenylacryloyl}amino)benzoate
ethyl 4-{[(2-hydroxy-3-iodo-6,7,8,9-tetrahydrodibenzo[b,d]furan-1-yl)methyl]amino}benzoate
2-({[4-ethyl-5-(4-pyridinyl)-4H-1,2,4-triazol-3-yl]sulfanyl}methyl)-6,7-dimethoxy-4(3H)-quinazolinone
ethyl 5-(3-methoxyanilino)[1,2,3]triazolo[1,5-a]quinazoline-3-carboxylate
ethyl 2-anilino-5-[(7-ethyl-1H-indol-3-yl)methylene]-4-oxo-4,5-dihydro-3-thiophenecarboxylate
ethyl 2-{[3-(aminocarbonyl)-4,5,6,7-tetrahydro-1-benzothien-2-yl]amino}-2-[(ethoxycarbonyl)amino]-3,3,3-trifluoropropanoate
ethyl 4-[(2,5-dimethyl-1-phenyl-1H-pyrrol-3-yl)methylene]-1-(2-methoxyethyl)-2-methyl-5-oxo-4,5-dihydro-1H-pyrrole-3-carboxylate
ethyl 2-[(2-fluorobenzoyl)amino]-4-isobutyl-3-thiophenecarboxylate
ethyl 2-({[2-(3-methoxyphenyl)-4-quinolinyl]carbonyl}amino)-4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-3-carboxylate
ethyl 2-{[2-(2,4-dichlorophenoxy)propanoyl]amino}-4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-3-carboxylate
2-[(4-ethyl-1-piperazinyl)carbonyl]benzoicacid
2-(4-ethylphenyl)-N-(1,3-thiazol-2-yl)-4-quinolinecarboxamide
ethyl 4-({6-[5-(4-chlorobenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]hexanoyl}amino)benzoate
ethyl 4-{[({5-[(2,4-dimethylanilino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}sulfanyl)acetyl]amino}benzoate
ethyl 4-(4-{[3,4-dimethyl(methylsulfonyl)anilino]methyl}benzoyl)piperazine-1-carboxylate
ethyl 4-(4-tert-butylphenyl)-2-{[(2,4-dichlorophenoxy)acetyl]amino}-3-thiophenecarboxylate
ethyl 5-(4-ethoxyphenyl)-7-methyl-3-oxo-2-(3-pyridinylmethylene)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
2-(ethylsulfanyl)ethyl 7-(3,4-dimethoxyphenyl)-4-(4-hydroxyphenyl)-2-methyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl 4-[({[1-(2,6-dimethylphenyl)-1H-tetraazol-5-yl]sulfanyl}acetyl)amino]benzoate
ethyl ({7-[2-hydroxy-3-(4-methoxyphenoxy)propyl]-3-methyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl}sulfanyl)acetate
ethyl 4-[5-({2,4-dioxo-3-[2-oxo-2-(1-pyrrolidinyl)ethyl]-1,3-thiazolidin-5-ylidene}methyl)-2-furyl]benzoate
ethyl 3-[({[4-(4-methoxyphenyl)-5-(4-toluidinomethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]benzoate
ethyl {2-[(4-iodobenzoyl)amino]-1,3-thiazol-4-yl}acetate
ethyl 3-amino-4-chloro-1-benzothiophene-2-carboxylate
ethyl 2-[(methoxycarbonyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
ethyl 4-(3-bromo-4,5-dimethoxyphenyl)-7-(3,4-dimethoxyphenyl)-2-methyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
2-ethyl-N-(4-methoxyphenyl)butanamide
3-ethyl-2-(ethylimino)-5-(1H-indol-3-ylmethylene)-1,3-thiazolidin-4-one
4-ethyl-5-(2-pyridinyl)-4H-1,2,4-triazol-3-yl 4-methylbenzyl sulfide
ethyl 2-{[2-(2,4-dichlorophenoxy)propanoyl]amino}-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
ethyl 5-({[(5-methyl-5H-[1,2,4]triazino[5,6-b]indol-3-yl)sulfanyl]acetyl}amino)-1-phenyl-1H-pyrazole-4-carboxylate
ethyl 4-(2-methoxybenzylidene)-2-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-pyrrole-3-carboxylate
3-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-N-[1-(4-fluorobenzyl)-1H-pyrazol-4-yl]acrylamide
ethyl 2-cyano-4-(1-[2-(4-methylphenyl)-2-oxoethyl]-4(1H)-quinolinylidene)-2-butenoate
ethyl 4-(1,3-benzodioxol-5-yl)-2-oxo-6-propyl-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate
ethyl 4-[(1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzoate
ethyl 5-(3-hydroxybenzylidene)-2-methyl-4-oxo-4,5-dihydro-1H-pyrrole-3-carboxylate
ethyl 6-amino-4-{5-[(4-bromophenoxy)methyl]-2,4-dimethylphenyl}-5-cyano-2-methyl-4H-pyran-3-carboxylate
2-{4-[(1-ethyl-1H-benzimidazol-2-yl)methyl]-1-piperazinyl}ethanol
2-ethyl-N-(2-pyridinylmethyl)hexanamide
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