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1-{[(4-ethyl-5-{[(4-fluorobenzyl)sulfanyl]methyl}-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-4-phenylpiperazine
5-ethyl-5-methyl-2-thioxo-2,3,5,6-tetrahydrobenzo[h]quinazolin-4(1H)-one
3-ethyl-5-nitroso-2-thioxo-1,3-thiazolidin-4-one
ethyl [(3-butyl-4-oxo-3,5,6,7-tetrahydro-4H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-2-yl)sulfanyl]acetate
ethyl 2-({2-[4-methoxy(methylsulfonyl)anilino]propanoyl}amino)benzoate
ethyl 2-(3-aminophenyl)-1,3-dioxo-5-isoindolinecarboxylate
ethyl 5-[4-(acetyloxy)phenyl]-2-[4-(diethylamino)benzylidene]-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
2-{[4-ethyl-5-(4-toluidinomethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(2-methoxyphenyl)acetamide
ethyl 6-amino-5-cyano-2-methyl-4-(3-methyl-2-thienyl)-4H-pyran-3-carboxylate
ethyl 2-(2,5-dimethoxybenzylidene)-5-(2-methoxy-1-naphthyl)-3-oxo-7-propyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 5-(benzoyloxy)-4-oxo-1,3-diphenyl-2-thioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidine-6-carboxylate
ethyl 2-[(3-bromobenzoyl)amino]-5-methyl-3-thiophenecarboxylate
ethyl 3-[({[5-methyl-4-(tetrahydro-2-furanylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]benzoate
ethyl 8-chloro-4-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-3-quinolinecarboxylate
ethyl 2-[({[3-(anilinomethyl)-1H-1,2,4-triazol-5-yl]sulfanyl}acetyl)amino]-4,5-dimethyl-3-thiophenecarboxylate
ethyl 2-[3-(2-furoyl)-4-hydroxy-2-(4-methylphenyl)-5-oxo-2,5-dihydro-1H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
ethyl 2-{4-[(2-chloro-6-fluorobenzyl)oxy]-3-methoxybenzylidene}-7-methyl-3-oxo-5-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 3-amino-4-(4-chlorophenyl)-6,7-dihydro-5H-cyclopenta[b]thieno[3,2-e]pyridine-2-carboxylate
ethyl 4-(4-chlorophenyl)-2-(pentanoylamino)-3-thiophenecarboxylate
ethyl 2-[4-(2-furoyloxy)-3-methoxybenzylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 3-[(5-chloro-2-methoxyanilino)carbonyl]-2-[(2-fluorobenzoyl)amino]-4,7-dihydrothieno[2,3-c]pyridine-6(5H)-carboxylate
ethyl 6-amino-5-cyano-2-(2-ethoxy-2-oxoethyl)-4-(2-methoxyphenyl)-4H-pyran-3-carboxylate
ethyl 6-amino-5-cyano-2-{[(3-cyano-6-phenyl-2-pyridinyl)sulfanyl]methyl}-4-(2-thienyl)-4H-pyran-3-carboxylate
ethyl 3-[(4-bromoanilino)carbonyl]-1-methyl-1H-pyrazole-5-carboxylate
ethyl (4-{[(4-methoxybenzyl)amino]sulfonyl}phenoxy)acetate
ethyl 2-({[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]acetyl}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl (2-amino-1,3-benzothiazol-6-yl)acetate
2-(4-ethylphenyl)-2-oxoethyl 4-[(phenylsulfonyl)amino]benzoate
ethyl 2-[(3-fluorobenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 5-[4-(acetyloxy)phenyl]-2-[4-(dimethylamino)benzylidene]-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 3-amino-2-(anilinocarbonyl)-4-(4-chlorophenyl)-6-methylthieno[2,3-b]pyridine-5-carboxylate
ethyl 5-(4-bromophenyl)-2-{[5-(dimethylamino)-2-furyl]methylene}-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl (9S)-9,10-dimethyl-11-thioxo-8-oxa-10,12-diazatricyclo[7.3.1.0~2,7~]trideca-2,4,6-triene-13-carboxylate
ethyl 4-({[2,5-dimethyl(methylsulfonyl)anilino]acetyl}amino)benzoate
ethyl 3,3,3-trifluoro-2-[(5-methyl-3-isoxazolyl)amino]-2-[(phenylacetyl)amino]propanoate
ethyl 4-methyl-5-({[4-(methyloxy)phenyl]amino}carbonyl)-2-[(phenylacetyl)amino]thiophene-3-carboxylate
ethyl 2-[(2,4-dichlorobenzoyl)amino]-3,3,3-trifluoro-2-[4-(trifluoromethyl)anilino]propanoate
ethyl 2-(5-bromo-3-ethoxy-2-hydroxybenzylidene)-7-methyl-3-oxo-5-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 6-tert-butyl-2-[(2-pyrazinylcarbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
4-ethylphenyl benzenesulfonate
ethyl 2-{[(3-cyano-5,6,7,8-tetrahydro-2-quinolinyl)sulfanyl]methyl}benzoate
ethyl 6-ethoxy-3-hydroxy-2-oxo-7-phenyl-2,5-dihydro-1H-azepine-4-carboxylate
ethyl 2-{[3-cyano-4,6-bis(4-methoxyphenyl)-2-pyridinyl]sulfanyl}acetate
ethyl 5-[4-(acetyloxy)-3-methoxyphenyl]-2-{[5-(2,4-dichlorophenyl)-2-furyl]methylene}-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
1-ethyl-3,6-diazatricyclo[4.3.1.1~3,8~]undecan-9-one oxime
3-(4-ethylphenyl)-2-[(4-ethylphenyl)imino]-5-[2-(hexyloxy)benzylidene]-1,3-thiazolidin-4-one
ethyl 2-[(9H-xanthen-9-ylcarbonyl)amino]-4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-3-carboxylate
ethyl 2-[5-nitro-2-(4-methyl-1-piperazinyl)benzylidene]-7-methyl-3-oxo-5-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-[(2-chlorobenzoyl)amino]-5-nitro-4-phenyl-3-thiophenecarboxylate
ethyl 3-(2-chloro-5-cyano-1,4-dimethyl-6-oxo-1,6-dihydro-3-pyridinyl)acrylate
ethyl 7-methyl-5-phenylpyrazolo[1,5-a]pyrimidine-2-carboxylate
ethyl 5-(4-chlorophenyl)-7-methyl-2-[(1-methyl-1H-pyrazol-4-yl)methylene]-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-{[(3-methyl-5-oxo-1-phenyl-1,5-dihydro-4H-pyrazol-4-ylidene)methyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 4-(2,3-dimethylphenyl)-1-piperazinecarboxylate
ethyl 4-({2,5-dimethoxy[(4-methylphenyl)sulfonyl]anilino}acetyl)piperazine-1-carboxylate
2-(4-ethylphenoxy)-N-[2-(4-morpholinylcarbonyl)phenyl]propanamide
ethyl 5-[(2-ethoxy-2-oxoethyl)sulfanyl]-3-methyl-1-phenyl-1H-thieno[2,3-c]pyrazole-4-carboxylate
ethyl 4-{2-nitrophenyl}-6-methyl-2-oxo-1-phenyl-1,2,3,4-tetrahydropyrimidine-5-carboxylate
ethyl 3-{[(2-(4-chlorophenyl)-5-oxo-1,3-oxazol-4(5H)-ylidene)methyl]amino}benzoate
ethyl 2-({[5-(2-furyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]carbonyl}amino)-4,5-dimethyl-3-thiophenecarboxylate
ethyl 2-({[2-(3,4-dichlorophenyl)-4-quinolinyl]carbonyl}amino)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 4-(2,3-dibromo-5-ethoxy-4-methoxyphenyl)-6-phenyl-2-thioxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate
4-ethyl 2-methyl 3-methyl-5-{[(1-methyl-1H-pyrazol-5-yl)carbonyl]amino}-2,4-thiophenedicarboxylate
ethyl 4-(4-ethoxy-3-methoxyphenyl)-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl 2-{[5-(3-chlorophenyl)-2-furyl]methylene}-7-methyl-3-oxo-5-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
3-ethyl-2-sulfanyl-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3H)-one
ethyl 4-[({[4-allyl-5-(4,5,6,7-tetrahydro-1-benzothien-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)amino]benzoate
ethyl 6-tert-butyl-2-({[2-(4-isopropoxyphenyl)-4-quinolinyl]carbonyl}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
2-ethyl-N-[3-(methylsulfanyl)phenyl]hexanamide
ethyl 2-({[3-(2,2-dichlorovinyl)-2,2-dimethylcyclopropyl]carbonyl}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 2-[({[(2-phenyl-4-quinolinyl)carbonyl]amino}carbothioyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 2-amino-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-7,7-dimethyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl (2-chloro-4-{[1-(4-fluorobenzyl)-2,5-dioxoimidazolidin-4-ylidene]methyl}-6-methoxyphenoxy)acetate
3-ethyl-5-[(5-morpholin-4-yl-2-furyl)methylene]-1,3-thiazolidine-2,4-dione
ethyl 2-[3-bromo-4-(dimethylamino)benzylidene]-3-oxo-7-phenyl-5-(2-thienyl)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
5-(1-ethyl-6-methyl-2(1H)-quinolinylidene)-1,3-dimethyl-2-thioxo-4-imidazolidinone
ethyl 4-{3-[(2-bromo-4-chlorophenoxy)methyl]-4-methoxyphenyl}-2-methyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl 6-amino-4-[2-chloro-6-(ethyloxy)quinolin-3-yl]-5-cyano-2-methyl-4H-pyran-3-carboxylate
ethyl 5-methyl-2-[(4-methyl-1-piperazinyl)methyl]-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-6-carboxylate
ethyl 4-[2-(difluoromethoxy)phenyl]-6-methyl-2-thioxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate
ethyl 5-(4-fluorophenyl)-2-(4-isopropylbenzylidene)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
2-({5-ethyl-4-nitro-2-thienyl}methylene)malononitrile
ethyl 4-{[(4-bromophenyl)acetyl]amino}benzoate
ethyl [(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]acetate
ethyl [2-({2-[(4-chlorophenyl)imino]-3-methyl-4-oxo-1,3-thiazolidin-5-ylidene}methyl)phenoxy]acetate
2-(4-ethylphenyl)-N-(4-isopropylphenyl)-4-quinolinecarboxamide
2-[4-ethyl(methylsulfonyl)anilino]-N-propylacetamide
ethyl 3-oxo-2-{[(4H-1,2,4-triazol-4-ylamino)carbothioyl]sulfanyl}butanoate
ethyl 5-acetyl-2-({[3-amino-4,6-bis(4-methoxyphenyl)thieno[2,3-b]pyridin-2-yl]carbonyl}amino)-4-methyl-3-thiophenecarboxylate
2-[2-ethyl(methylsulfonyl)anilino]-N-[4-(1-pyrrolidinylsulfonyl)phenyl]acetamide
3-ethyl-2-[(4-ethylphenyl)imino]-5-(2-hydroxybenzylidene)-1,3-thiazolidin-4-one
ethyl 5-phenyl-2-{[(4-phenyl-1-piperazinyl)acetyl]amino}-3-thiophenecarboxylate
ethyl 2-{[3-cyano-6-(4-ethoxyphenyl)-4-phenyl-2-pyridinyl]sulfanyl}butanoate
ethyl 2-({[(1-methyl-1H-imidazol-2-yl)sulfanyl]acetyl}amino)-5-phenyl-3-thiophenecarboxylate
ethyl 2-{[3-cyano-6-(2-furyl)-4-(trifluoromethyl)pyridin-2-yl]sulfanyl}propanoate
ethyl 5-{4-nitrophenyl}-1,3,4-thiadiazol-2-ylcarbamate
1-ethyl-N-[2-(phenylsulfanyl)phenyl]-1H-pyrazole-3-carboxamide
ethyl 2-(1-benzoyl-2,2-dimethyl-3-thioxo-2,3-dihydro-4(1H)-quinolinylidene)-5-phenyl-1,3-dithiole-4-carboxylate
ethyl (3-thioxo-1,2,4-triazaspiro[4.7]dodec-2-yl)acetate
ethyl 4-cyano-5-({[2-(2,4-dimethoxyphenyl)-4-quinolinyl]carbonyl}amino)-3-methyl-2-thiophenecarboxylate
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