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ethyl 2-{4-nitrobenzylidene}-7-methyl-3-oxo-5-(2-phenylvinyl)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 3-[(3-chloro-4-methylbenzoyl)amino]-4-(4-morpholinyl)benzoate
ethyl 2-[(8-{[3-(ethoxycarbonyl)-5,6-dihydro-4H-cyclopenta[b]thien-2-yl]amino}-8-oxooctanoyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
ethyl 2-(benzoylamino)-5-[(3-chloroanilino)carbonyl]-4-methylthiophene-3-carboxylate
ethyl 1-({(3-chlorobenzyl)[(4-methylphenyl)sulfonyl]amino}acetyl)piperidine-4-carboxylate
ethyl 2-[(3-ethyl-4,8-dimethyl-2-oxo-2H-chromen-7-yl)oxy]propanoate
ethyl 4-{4-[(4-chlorophenoxy)methyl]-5-methyl-2-thienyl}-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl 2-{3-ethoxy-4-[(2-iodobenzoyl)oxy]benzylidene}-7-methyl-3-oxo-5-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
3-ethyl-5-{[3-(4-ethylphenyl)-1H-pyrazol-4-yl]methylene}-2-thioxo-1,3-thiazolidin-4-one
ethyl 2-amino-4-(4-methoxy-3-{[3-(trifluoromethyl)phenoxy]methyl}phenyl)-5-oxo-5,6,7,8-tetrahydro-4H-chromene-3-carboxylate
ethyl 5-[4-(dimethylamino)phenyl]-7-methyl-3-oxo-2-[(1,3,5-trimethyl-1H-pyrazol-4-yl)methylene]-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-(1-naphthylamino)-4-oxo-4,5-dihydrothiophene-3-carboxylate
ethyl {4-[(1,3-benzodioxol-5-ylamino)sulfonyl]phenoxy}acetate
ethyl 2-(4-methoxyanilino)-4-oxo-5-(1H-pyrrol-2-ylmethylene)-4,5-dihydro-3-thiophenecarboxylate
ethyl 2-{5-[(6-ethoxy-1,3-benzodioxol-5-yl)methylene]-2,4-dioxo-1,3-thiazolidin-3-yl}propanoate
ethyl 2-{[4-(difluoromethoxy)-3-methoxybenzoyl]amino}-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
ethyl 4-{[2-[(1-adamantylcarbonyl)amino]-3-(1H-indol-3-yl)propanoyl]amino}benzoate
4-ethyl-N-(3-methoxyphenyl)benzamide
ethyl 2-{[5-(4-bromophenyl)-2-furyl]methylene}-5-(2-chlorophenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 4-[4-(allyloxy)-3-iodo-5-methoxyphenyl]-6-amino-5-cyano-2-methyl-4H-pyran-3-carboxylate
ethyl pyrrolo[1,2-c]quinazoline-2-carboxylate
ethyl 2-(4-chlorobenzylidene)-7-methyl-5-(4-methylphenyl)-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-[(4-{4-chloro-3-nitro-5-methyl-1H-pyrazol-1-yl}butanoyl)amino]-4,5-dimethyl-3-thiophenecarboxylate
ethyl 6-methyl-2-({[(5-methyl[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]acetyl}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
3-[(2-ethylhexanoyl)amino]-N-(4-methyl-2-pyridinyl)benzamide
5-(ethylsulfonyl)-1,3-benzoxazol-2-yl hydrosulfide
ethyl 2-({[(4-methyl-2-pyridinyl)amino]carbothioyl}amino)-5-phenyl-3-thiophenecarboxylate
ethyl 1,6-dimethyl-4-(5-methyl-2-thienyl)-2-oxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate
ethyl (5-{[1-(1,3-benzodioxol-5-yl)-2,5-dimethyl-1H-pyrrol-3-yl]methylene}-2,4-dioxo-1,3-thiazolidin-3-yl)acetate
ethyl 2,4-bis[(2-oxopropyl)sulfanyl]-5,8-dihydropyrido[4',3':4,5]thieno[2,3-d]pyrimidine-7(6H)-carboxylate
ethyl 4-({[(2-fluorobenzoyl)amino]carbothioyl}amino)benzoate
ethyl 2-{[3-cyano-6-(4-methylphenyl)-4-phenyl-2-pyridinyl]sulfanyl}propanoate
ethyl 5-(4-chlorophenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxylate
ethyl 2-{2-[(4-chlorobenzyl)oxy]benzylidene}-5-(2-methoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
7-[3-(4-ethylphenoxy)-2-hydroxypropyl]-3-methyl-8-(octylsulfanyl)-3,7-dihydro-1H-purine-2,6-dione
ethyl 5-(acetyloxy)-2-({[anilino(imino)methyl]sulfanyl}methyl)-6-bromo-1-(4-methylphenyl)-1H-indole-3-carboxylate
ethyl 2-anilino-4-oxo-5-({1-[2-oxo-2-(1-pyrrolidinyl)ethyl]-1H-indol-3-yl}methylene)-4,5-dihydro-3-thiophenecarboxylate
6-ethyl-N-(4-methoxyphenyl)-2-phenyl-4-quinolinecarboxamide
ethyl 5-[(5-ethyl-2-thienyl)methylene]-2-[(4-methylbenzoyl)amino]-4-oxo-4,5-dihydro-3-thiophenecarboxylate
2-{[4-ethyl-5-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N'-(4-methoxybenzoyl)acetohydrazide
ethyl 2-{[3-(trifluoromethyl)benzoyl]amino}-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
ethyl 3-amino-4-(2-furyl)-6-phenylfuro[2,3-b]pyridine-2-carboxylate
1-ethyl-N-(2-fluoro-5-methylphenyl)-4-nitro-1H-pyrazole-3-carboxamide
ethyl 2-{2-[2-(benzylamino)-2-oxoethoxy]benzylidene}-5-(4-hydroxy-3-methoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl7-{4-[(2-fluorobenzyl)oxy]-3-methoxyphenyl}-5-methyl-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
ethyl 4-(aminocarbonyl)-5-({[2-(4-ethoxyphenyl)-4-quinolinyl]carbonyl}amino)-3-methyl-2-thiophenecarboxylate
ethyl [4-({3-[2-(4-morpholinyl)-2-oxoethyl]-2,4-dioxo-1,3-thiazolidin-5-ylidene}methyl)phenoxy]acetate
ethyl 4-[({4-chloro-2-nitrophenyl}carbonyl)amino]benzoate
ethyl (5-{[5-(4-bromo-3-chlorophenyl)-2-furyl]methylene}-2,4-dioxo-1,3-thiazolidin-3-yl)acetate
ethyl 5-(aminocarbonyl)-1-methyl-1H-pyrazole-3-carboxylate
2-[(4-ethyl-5-pyridin-3-yl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-phenylacetamide
ethyl 2-{[phenyl(phenylsulfanyl)acetyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl [(ethoxycarbonyl)amino](3-ethoxy-4-methoxyphenyl)methylcarbamate
ethyl 2-(2-hydroxy-3-methoxybenzylidene)-7-methyl-5-(4-methylphenyl)-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 6-bromo-2-(chloromethyl)-5-methoxy-1-methyl-1H-indole-3-carboxylate
ethyl 2-(4-fluorobenzylidene)-5-(2-methoxyphenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
1-ethyl-4-nitro-N-[5-methyl-4-(4-methylphenyl)-1,3-thiazol-2-yl]-1H-pyrazole-3-carboxamide
ethyl 2-(methylsulfanyl)-4-{[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]sulfanyl}-5-pyrimidinecarboxylate
2-(ethylsulfanyl)ethyl 4-(3-ethoxyphenyl)-6-methyl-2-oxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate
ethyl 2-tert-butyl-5-[(2-methylbenzoyl)oxy]-1-benzofuran-3-carboxylate
ethyl 5-amino-6-cyano-2-{3-nitrobenzylidene}-7-{3-nitrophenyl}-3-oxo-2,3-dihydro-7H-[1,3]thiazolo[3,2-a]pyridine-8-carboxylate
ethyl 5-(4-isopropoxyphenyl)-7-methyl-3-oxo-2-(2-pyridinylmethylene)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 5-[4-(dimethylamino)phenyl]-7-methyl-2-{[5-(4-morpholinyl)-2-furyl]methylene}-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 5-(4-fluorophenyl)-2-[5-nitro-2-(1-piperidinyl)benzylidene]-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
ethyl 2-({[(3-allyl-4-oxo-3,5,6,7,8,9-hexahydro-4H-cyclohepta[4,5]thieno[2,3-d]pyrimidin-2-yl)sulfanyl]acetyl}amino)-4-(2-furyl)-3-thiophenecarboxylate
ethyl 2-amino-7,7-dimethyl-5-oxo-1-[2-(trifluoromethyl)phenyl]-4-(3,4,5-trimethoxyphenyl)-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl [(5-sulfanyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetate
ethyl 5-[(benzylamino)carbonyl]-4-methyl-2-[(2-thienylcarbonyl)amino]-3-thiophenecarboxylate
ethyl [2-({2-[(4-methylphenyl)imino]-4-oxo-1,3-thiazolidin-5-ylidene}methyl)phenoxy]acetate
ethyl 8-chloro-4-{3-nitroanilino}-3-quinolinecarboxylate
ethyl 2-[3-chloro-5-ethoxy-4-(2-propynyloxy)benzylidene]-5-(4-fluorophenyl)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
7-{[{[(4-ethyl-2,3-dioxo-1-piperazinyl)carbonyl]amino}(4-hydroxyphenyl)acetyl]amino}-3-{[(1-methyl-1H-tetraazol-5-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate
ethyl ([1]benzofuro[3,2-d]pyrimidin-4-ylsulfanyl)acetate
ethyl 4-benzoyl-1-(4-ethoxyphenyl)-5-phenyl-1H-pyrazole-3-carboxylate
ethyl 4-(3-bromophenyl)-2-[(pyrazin-2-ylcarbonyl)amino]thiophene-3-carboxylate
ethyl 5-[3-ethoxy-4-(2-methoxy-2-oxoethoxy)benzylidene]-4-oxo-2-(4-toluidino)-4,5-dihydro-3-thiophenecarboxylate
ethyl 5-{butyryl[(2,5-dimethylphenyl)sulfonyl]amino}-2-methyl-1-benzofuran-3-carboxylate
ethyl 4-{[3-(4-methoxyphenyl)-4-phenyl-5-thioxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}-1-piperazinecarboxylate
ethyl 4-(5-tert-butyl-2-thienyl)-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydro-3-quinolinecarboxylate
ethyl ({2-[(3-bromobenzoyl)amino]-3-phenylacryloyl}amino)acetate
ethyl 4-{[[(3-hydroxypropyl)amino](oxo)acetyl]amino}benzoate
ethyl 1,6-dimethyl-2-phenyl-4-thioxo-1,4-dihydro-5-pyrimidinecarboxylate
ethyl 2-[(2-methoxybenzoyl)amino]-5-methyl-4-(4-methylphenyl)-3-thiophenecarboxylate
ethyl 2-[(2-methoxybenzoyl)amino]-5-phenylthiophene-3-carboxylate
ethyl 5-(4-methylphenyl)-3-[(1-pyrrolidinylcarbothioyl)amino]-2-thiophenecarboxylate
ethyl 3-({[(4,5-dimethyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}amino)benzoate
ethyl 6-amino-5,7,7-tricyano-8-[2-(trifluoromethyl)phenyl]-3,7,8,8a-tetrahydro-2(1H)-isoquinolinecarboxylate
ethyl 4-amino-6-methyl-2-phenyl-5-pyrimidinecarboxylate
ethyl 2-({[5-(4-methylbenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetyl}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
ethyl 9-[2-(diethylamino)ethyl]-2-methyl-9H-imidazo[1,2-a]benzimidazole-3-carboxylate
ethyl 2-(4-{[(diethoxyphosphoryl)(4-methoxyphenyl)methyl]amino}phenyl)-3,3,3-trifluoro-2-hydroxypropanoate
ethyl 4-({[4-chloro(phenylsulfonyl)anilino]acetyl}amino)benzoate
ethyl ethoxy(phenyl)methylcarbamate
2-[(2-ethylbutanoyl)amino]benzamide
ethyl 2-{[3-cyano-4-(4-methoxyphenyl)-6-phenyl-2-pyridinyl]sulfanyl}butanoate
ethyl 2-{[(2-chlorophenyl)acetyl]amino}-5-ethyl-3-thiophenecarboxylate
ethyl 2-({[3-(2-chlorophenyl)-5-methyl-4-isoxazolyl]carbonyl}amino)-4-ethyl-5-methyl-3-thiophenecarboxylate
1-ethyl-3-hydroxy-3-(2-oxo-4-phenyl-3-butenyl)-1,3-dihydro-2H-indol-2-one
ethyl 5-(4-isopropoxyphenyl)-7-methyl-3-oxo-2-(2-thienylmethylene)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
2-(ethylsulfanyl)-9-oxo-4-(2-thienyl)-9H-indeno[2,1-b]pyridine-3-carbonitrile
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